MUC1 & CD28
This gene encodes a membrane-bound protein that is a member of the mucin family. Mucins are O-glycosylated proteins that play an essential role in forming protective mucous barriers on epithelial surfaces. These proteins also play a role in intracellular signaling. This protein is expressed on the apical surface of epithelial cells that line the mucosal surfaces of many different tissues including lung, breast stomach and pancreas. This protein is proteolytically cleaved into alpha and beta subunits that form a heterodimeric complex. The N-terminal alpha subunit functions in cell-adhesion and the C-terminal beta subunit is involved in cell signaling. Overexpression, aberrant intracellular localization, and changes in glycosylation of this protein have been associated with carcinomas. This gene is known to contain a highly polymorphic variable number tandem repeats (VNTR) domain. Alternate splicing results in multiple transcript variants.
Enables protein kinase binding activity. Acts upstream of or within several processes, including positive regulation of immune response; positive regulation of intracellular signal transduction; and regulation of lymphocyte activation. Located in external side of plasma membrane and immunological synapse. Human ortholog(s) of this gene implicated in multiple sclerosis and type 1 diabetes mellitus. Orthologous to human CD28 (CD28 molecule).
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- Targets: MUC1 & CD28
- Type: Fab2
- Application: FuncS, Promising therapeutic agent
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- Species Reactivity: Human, Non-Human Primates
- Type: Mouse IgG1
- Application: FC, IP, WB, IHC, FuncS
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- Derivation: Mouse
- Species Reactivity: Canine
- Type: Mouse scFv
- Application: WB, ELISA, FuncS
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- Derivation: Mouse
- Species Reactivity: canine
- Type: Mouse IgG1
- Application: WB, ELISA, FuncS
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- Derivation: Mouse
- Species Reactivity: Human
- Type: Mouse IgG1, κ
- Application: WB, FC, IF, IHC
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- Derivation: Mouse
- Species Reactivity: Human
- Type: Mouse IgG
- Application: WB, IF, FuncS
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- Derivation: Mouse
- Species Reactivity: canine
- Type: Mouse Fab
- Application: WB, ELISA, FuncS
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- Derivation: Mouse
- Species Reactivity: Human
- Type: Mouse scFv
- Application: WB, IF, FuncS
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- Derivation: Mouse
- Species Reactivity: Human
- Type: Mouse Fab
- Application: WB, IF, FuncS
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- Target: CanAg
- Linker: SPDB(N-succinimidyl 4-(2-pyridyldithio)butyrate)
- Drug: [3H]DM4([3H]N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Species Reactivity: Human
- Type: Mouse IgG
- Application: FC, ELISA, IF
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- Host Species: Human
- Specificity: Human
- Type: Humanized antibody
- Glycosylation site: CDR2 of VH
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- Species Reactivity: Human
- Type: Mouse Fab
- Application: ELISA, SDS-PAGE, IHC
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: FC, ELISA, IF
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- Species Reactivity: Human
- Type: Mouse IgG
- Application: FC, ELISA, IF
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- Host Species: Human
- Specificity: Human
- Type: Humanized antibody
- Glycosylation site: CDR2 of VH
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- Species Reactivity: Human
- Type: Mouse Fab
- Application: ELISA, SDS-PAGE, IHC
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: ELISA, IHC
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- Species Reactivity: Human
- Type: Mouse IgG
- Application: ELISA, IHC, WB
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- Species Reactivity: Human
- Type: Mouse Fab
- Application: IF
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: ELISA, SDS-PAGE, IHC
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- Species Reactivity: Human
- Type: Mouse IgG1
- Application: ELISA, IHC, IF, FC
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- Species Reactivity: Human
- Type: Mouse Fab
- Application: IF
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: FC, ELISA
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: ELISA, SDS-PAGE, IHC
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- Species Reactivity: Human
- Type: Mouse IgG1
- Application: ELISA, FuncS, IHC, IF, FC, ADCC
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- Species Reactivity: Human
- Type: Humanized Fab
- Application: ELISA
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: FC, ELISA
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: IF
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- Species Reactivity: Human
- Type: Mouse IgG
- Application: IF
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- Species Reactivity: Human
- Type: Chimeric (mouse/human) Fab
- Application: ELISA
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: FC, ELISA
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: IF
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- Species Reactivity: Human
- Type: Mouse IgG
- Application: Block
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- Species Reactivity: Human
- Type: Mouse Fab
- Application: ELISA
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: FC, ELISA
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- Species Reactivity: Human
- Type: Humanized scFv
- Application: ELISA
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- Species Reactivity: Human
- Type: Humanized IgG
- Application: ELISA
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- Derivation: Humanized
- Type: Humanized antibody
- Application: FC, ELISA
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- Species Reactivity: Human
- Type: Human scFv
- Application: ELISA, FC
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: ELISA
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- Species Reactivity: Human
- Type: Chimeric (mouse/human) IgG
- Application: ELISA
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- Derivation: Chimeric (mouse/human)
- Type: Chimeric antibody (mouse/human)
- Application: FC, ELISA
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- Derivation: Humanized
- Type: Humanized antibody
- Application: ELISA, FC
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- Species Reactivity: Human
- Type: Mouse scFv
- Application: ELISA
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- Species Reactivity: Human
- Type: Mouse IgG
- Application: ELISA
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- Derivation: Humanized
- Species Reactivity: Human
- Type: Humanized Fab
- Application: ELISA
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- Derivation: Chimeric (mouse/human)
- Type: Chimeric antibody (mouse/human)
- Application: ELISA, FC
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- Derivation: Humanized
- Species Reactivity: Human
- Type: Humanized Fab
- Application: ELISA
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- Derivation: Humanized
- Species Reactivity: Human
- Type: Human IgG1
- Application: FC, IF, ELISA
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- Derivation: Humanized
- Type: Humanized antibody
- Application: FC, ELISA
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- Derivation: Humanized
- Species Reactivity: Human
- Type: Human IgG, κ
- Application: ELISA
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- Derivation: Humanized
- Species Reactivity: Human
- Type: Human scFv
- Application: ELISA
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- Derivation: Chimeric (mouse/human)
- Type: Chimeric antibody (mouse/human)
- Application: FC, ELISA
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- Derivation: Humanized
- Type: Humanized antibody
- Application: FC
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- Derivation: Humanized
- Type: Humanized antibody
- Application: FC, Stim
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- Derivation: Humanized
- Species Reactivity: Human
- Type: Human scFv
- Application: ELISA
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- Derivation: Humanized
- Type: Humanized antibody
- Application: FC
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- Species Reactivity: Human
- Type: Human Fab
- Application: ELISA, Internalization, BI, FuncS
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- Target: mucin repeats
- Linker: VC (valine-citrulline)
- Drug: MMAF (monomethyl auristatin F)
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- Species Reactivity: Human
- Type: Human scFv
- Application: ELISA, Internalization, BI, FuncS
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- Target: mucin repeats
- Linker: mc (maleimidocaproyl)
- Drug: MMAF (monomethyl auristatin F)
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- Species Reactivity: Human
- Type: Human IgG
- Application: ELISA, Internalization, BI, FuncS
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- Target: CanAg
- Linker: SMCC (4-[N-maleimidomethyl] cyclohexane-1 carboxylhydrazide).
- Drug: [3H]DM1([3H]N2'-deacetyl-N2'-(3-mercapto-1-oxopropyl)-maytansine)
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- Species Reactivity: Human
- Type: Mouse IgG1 F(ab')2, κ
- Application: Agonist, Stim, Neu, FC
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- Species Reactivity: Human
- Type: Llama VHH
- Application: WB, IP, ChiP, Neut, ELISA
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- Target: CAIX, Carbonic anhydrase IX
- Linker: mcc (Maleimidomethyl cyclohexane-1-carboxylate)
- Drug: MMAE (Monomethyl auristatin E)
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- Target: CanAg
- Linker: SPP(N-succinimidyl 4-(2-pyridyldithio)pentanoate)
- Drug: [3H]DM1([3H]N2'-deacetyl-N2'-(3-mercapto-1-oxopropyl)-maytansine)
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- Derivation: Humanized
- Species Reactivity: Human
- Type: Humanized V-kappa
- Application: IP, IF, FuncS, FC, Neut, ELISA, IHC
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- Species Reactivity: Human
- Application: Cytotoxicity assay, Functional assay
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- Species Reactivity: Human
- Application: Cytotoxicity assay, Functional assay
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- Derivation: Humanized (from mouse)
- Species Reactivity: Human
- Type: Fab - G1 - kappa
- Application: Neut, ELISA, IF, IP, FuncS, FC, IHC
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- Derivation: Mouse
- Species Reactivity: Human
- Type: Mouse Fab (IgG1, κ)
- Application: FC, IP, ELISA, Neut, FuncS, IF, ICC
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- Derivation: Humanized (from mouse)
- Species Reactivity: Human
- Type: Humanized (from mouse) IgG1, κ
- Application: IP, IF, FuncS, FC, Neut, ELISA, ICC
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- Derivation: Humanized (from mouse)
- Species Reactivity: Human
- Type: IgG1 - kappa
- Application: IF, IP, Neut, FuncS, ELISA, FC, ICC
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- Target: CD28
- Species Reactivity: Human
- Cytokine 1: TNF
- Host: Mouse
- Cytokine 1 Species: Human
- Molecule Class: TNF-IgG2a
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- Target: CanAg
- Linker: SPP (N-succinimidyl-4-(2-pyridyldithio)pentanoate)
- Drug: DM1 (N2'-Deacetyl-N2'-(3-mercapto-1-oxopropyl)maytansine)
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- Target: CanAg
- Linker: SPDB(N-succinimidyl 4-(2-pyridyldithio)butyrate)
- Drug: DM4(N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Target: CD28
- Species Reactivity: Human
- Cytokine 1: IL2
- Host: Mouse
- Cytokine 1 Species: Human
- Molecule Class: IL2-IgG2a
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- Target: Mucin1
- Drug: DM4(N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Target: CanAg
- Linker: SPDB
- Drug: DM4 (N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Target: CanAg
- Linker: SMCC (4-[N-maleimidomethyl] cyclohexane-1 carboxylhydrazide).
- Drug: DM1(N2'-deacetyl-N2'-(3-mercapto-1-oxopropyl)-maytansine)
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- Target: MUC-1
- Species Reactivity: Human
- Cytokine 1: IL2
- Host: Chimeric (Human-Mouse)
- Cytokine 1 Species: Human
- Molecule Class: scFv-Fc-IL2
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- Target: CanAg
- Linker: SPDB (N-succinimidyl 4-(2-pyridyldithio)butyrate)
- Drug: DM4(N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Target: CanAg
- Linker: sulfo-SPDB (sulfo-N-succinimidyl 4-(2-pyridyldithio)butyrate
- Drug: DM4 (N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Target: CanAg
- Linker: SPP(N-succinimidyl 4-(2-pyridyldithio)pentanoate)
- Drug: DM1(N2'-deacetyl-N2'-(3-mercapto-1-oxopropyl)-maytansine)
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- Target: MUC1
- Linker: CL2A
- Drug: SN-38(7-ethyl-10-hydroxy camptothecin)
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- Target: CanAg
- Linker: SMCC (4-[N-maleimidomethyl] cyclohexane-1 carboxylhydrazide).
- Drug: DM1(N2'-deacetyl-N2'-(3-mercapto-1-oxopropyl)-maytansine)
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- Target: CanAg
- Linker: SMCC (N-succinimidyl 4-(Nmaleimidomethyl)cyclohexane-1-carboxylate)
- Drug: DM1 (N2'-Deacetyl-N2'-(3-mercapto-1-oxopropyl)maytansine)
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- Derivation: Humanized (from mouse)
- Species Reactivity: Human
- Type: IgG1
- Application: WB, ELISA, FC, IP, FuncS, IF, Neut
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- Target: CanAg
- Linker: SPDB (N-succinimidyl 4-(2-pyridyldithio)butyrate)
- Drug: DM4(N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Target: CA6, a specific glycol-epitope of MUC-1
- Linker: SPDB (N-succinimidyl 4-(2-pyridyldithio)butyrate)
- Drug: DM4(N2'-Deacetyl-N2'-(4-mercapto-4-methyl-1-oxopentyl)maytansine)
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- Target: CanAg
- Linker: PEG4Mal
- Drug: DM1 (N2'-Deacetyl-N2'-(3-mercapto-1-oxopropyl)maytansine)
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- Derivation: Mouse
- Species Reactivity: Human
- Type: IgG
- Application: WB, FuncS, IF, Neut, ELISA, FC, IP
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- Derivation: Humanized
- Species Reactivity: Human
- Type: IgG1, κ
- Application: FuncS, Inhib
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- Target: mucin
- Drug: SN-38 (7-ethyl-10-hydroxycamptothecin)
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